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  • GSK1016790A

    2025-07-19

    GSK1016790A

    Author: ApexBio

    spu:

    C5065

    CAS:

    942206-85-1

    purity:

    0.9945

    shortsummary:

    TRPV4 agonist

    740y-p site

    Formula:

    C28H32Cl2N4O6S2

    M.Wt:

    655.6

    Chemical Name:

    N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbonyl]-3-methylbutyl]-benzo[b]thiophene-2-carboxamide

    SMILES:

    ClC1=CC=C(S(N[C@H](C(N2CCN(C([C@@H](NC(C3=CC4=C(C=CC=C4)S3)=O)CC(C)C)=O)CC2)=O)CO)(=O)=O)C(Cl)=C1

    Solubility:

    ≥50.4 mg/mL in DMSO; ≥26.3 mg/mL in EtOH; insoluble in H2O

    Storage:

    Store at -20°C

    Physical Appearance:

    A crystalline solid

    DeliveryTime:

    In stock

    740 Y-P supplier

    ShippingType:

    Blue ice

    description:

    GSK1016790A is a small molecule TRPV4 channel activator [1].

    GSK1016790A PMC11287020

    related websites:

    APExBIO Technology LLC is a premier provider of Small Molecule Inhibitors/Activators, Compound Libraries, Peptides, Assay Kits, Fluorescent Labels, Enzymes, Modified Nucleotides, mRNA synthesis and various tools for Molecular Biology. We carry a broad product line in over 16246 different research areas such as cancer, immunology, neurosciences, apoptosis and epigenetics etc. Based in USA (Houston, Texas), we have been serving the needs of customers across the world.

    https://www.apexbt.com/